Molecule Details
InChIKeyGMEWMQLWXBFPOI-ZJZDTXIUSA-N
Compound NameD-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe-Nle-NH2
Canonical SMILESCCCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](C)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](N)Cc1ccccc1)C(C)C)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32247 BRS3 Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P30550 GRPR Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P28336 NMBR Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB