Molecule Details
InChIKeyGMDLUFKQPDBUPT-FIFLTTCUSA-N
Compound NameN-hydroxy-3-(4-(3-(2-methoxyphenyl)-3-oxoprop-1-enyl)-1-methyl-1H-pyrrol-2-yl)acrylamide
Canonical SMILESCOc1ccccc1C(=O)/C=C/c1cc(/C=C/C(=O)NO)n(C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.77
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 6.8 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.8 pIC50 TTD_MultiTarget
Q92769 HDAC2 Homo sapiens Human PF00850 6.8 pIC50 TTD_MultiTarget