Molecule Details
InChIKeyGLCIBEGENZSGCS-UHFFFAOYSA-N
Compound Name2-(4-fluorophenyl)-N-[5-(4-pyridin-3-ylthiophen-2-yl)-3-pyridinyl]acetamide
Canonical SMILESO=C(Cc1ccc(F)cc1)Nc1cncc(-c2cc(-c3cccnc3)cs2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q8TF76 HASPIN Homo sapiens Human PF12330 7.4 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB