Molecule Details
InChIKeyGKWZHZVUJVOVJN-FQEVSTJZSA-N
Compound NameN-[(R)-(3,4-dichlorophenyl)-(1-methylazetidin-3-yl)methyl]isoquinoline-6-carboxamide
Canonical SMILESCN1CC([C@@H](NC(=O)c2ccc3cnccc3c2)c2ccc(Cl)c(Cl)c2)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P31749 AKT1 Homo sapiens Human PF00169 PF00069 PF00433 8.2 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget