Molecule Details
InChIKeyGKQWMOXIBZCMDJ-PWZOGDDVSA-N
Compound Name(6S,9S,10R,13S,14S,17R)-17-acetyl-6,10,13-trimethyl-17-(2-oxopropyl)-2,6,7,8,9,11,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthren-3-one
Canonical SMILESCC(=O)C[C@]1(C(C)=O)CC[C@H]2C3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@@]21C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 9.5 Ki ChEMBL;BindingDB
P10275 AR Homo sapiens Human PF02166 PF00104 PF00105 8.2 IC50 ChEMBL;BindingDB
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 8.0 IC50 ChEMBL;BindingDB