Molecule Details
InChIKeyGKODDLYLEKSDJL-UHFFFAOYSA-N
Canonical SMILESCCOc1nc(NC(=O)Cc2cc(OC)c(Br)cc2OC)cc(N)c1C#N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07272
Drug NameN-(4-AMINO-5-CYANO-6-ETHOXYPYRIDIN-2-YL)-2-(4-BROMO-2,5-DIMETHOXYPHENYL)ACETAMIDE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 15940 CHEMBL382639 ChemSpider: 5254658 PDB: 877 PubChem:6852206 PubChem:99443743 ZINC: ZINC000014960080
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P45983 MAPK8 Mitogen-activated protein kinase 8 binder targets
Q9UQF2 Q9UQF2 C-Jun-amino-terminal kinase-interacting protein 1 binder targets