Molecule Details
InChIKeyGJZGXWPLIMVUDJ-UHFFFAOYSA-N
Compound NameUS10221163, Example 12
Canonical SMILESNCCNS(=O)(=O)c1ccc(-c2cccc3[nH]c(N)nc23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.95
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.4 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 10.0 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.5 IC50 BindingDB