Molecule Details
InChIKeyGJTOCPGDDLTBBD-LHRJYYJOSA-N
Compound Name(2S)-N-[(2S,3S)-5-[[(2S)-1-[[(2S)-1-[[(2R)-1-(benzylamino)-1-oxo-3-phenylpropan-2-yl]-methylamino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-5-oxo-1-phenylpentan-2-yl]-2-[[(2S)-2-[[(2S)-2-hydroxypropanoyl]amino]-3-methylbutanoyl]-methylamino]pentanediamide
Canonical SMILESCC(C)C[C@H](NC(=O)C[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)N(C)C(=O)[C@@H](NC(=O)[C@H](C)O)C(C)C)C(=O)N[C@@H](C)C(=O)N(C)[C@H](Cc1ccccc1)C(=O)NCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07339 CTSD Homo sapiens Human PF07966 PF00026 7.7 IC50 ChEMBL;BindingDB
P14091 CTSE Homo sapiens Human PF07966 PF00026 7.5 IC50 ChEMBL;BindingDB
P56817 BACE1 Homo sapiens Human PF00026 6.9 IC50 ChEMBL;BindingDB