Molecule Details
InChIKeyGJRUPTCKZNHKDR-UKTHLTGXSA-N
Compound Name4-[(E)-(3-methyl-5-sulfamoyl-1,3,4-thiadiazol-2-ylidene)amino]sulfonylbenzoic acid
Canonical SMILESCn1nc(S(N)(=O)=O)s/c1=N/S(=O)(=O)c1ccc(C(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.95
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.3 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.3 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.3 Ki ChEMBL;BindingDB