Molecule Details
InChIKeyGJPQENHVEQGHGP-UMCMBGNQSA-N
Compound Namemethyl 6-[3-[[~{N}-[[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl]carbamimidoyl]amino]propylcarbamoylamino]-4-oxidanyl-naphthalene-2-carboxylate
Canonical SMILESCOC(=O)c1cc(O)c2cc(NC(=O)NCCCNC(=N)NC[C@H]3O[C@@H](n4cnc5c(N)ncnc54)[C@H](O)[C@@H]3O)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.24
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NVM4 PRMT7 Homo sapiens Human PF06325 PF22528 6.5 IC50 ChEMBL
Q86X55 CARM1 Homo sapiens Human PF11531 PF06325 PF22528 6.2 Kd ChEMBL
Q6P2P2 PRMT9 Homo sapiens Human PF06325 PF22528 6.0 IC50 ChEMBL