Molecule Details
InChIKeyGIXKBVCWMSZXME-UHFFFAOYSA-N
Compound Name7-[2-(Piperidin-4-yloxy)-carbazol-9-ylmethyl]-naphthalene-2-carboxamidine
Canonical SMILESN=C(N)c1ccc2ccc(Cn3c4ccccc4c4ccc(OC5CCNCC5)cc43)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 8.4 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.5 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.8 Ki ChEMBL;BindingDB