Molecule Details
InChIKeyGIQHYUIXZZZJQF-HXUWFJFHSA-N
Compound Name4-methyl-8-[3-[(2R)-2-methyl-4-(2-methylquinolin-5-yl)piperazin-1-yl]propyl]-1,4-benzoxazin-3-one
Canonical SMILESCc1ccc2c(N3CCN(CCCc4cccc5c4OCC(=O)N5C)[C@H](C)C3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 9.3 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB