Molecule Details
InChIKeyGIAAJPPEMQIXPQ-UHFFFAOYSA-N
Compound Name3-[3-[[2-[(4-chloro-1H-benzimidazol-5-yl)methyl-methylamino]pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]cyclopentan-1-one
Canonical SMILESCN(Cc1ccc2[nH]cnc2c1Cl)c1nccc(Nc2cc(C3CCC(=O)C3)[nH]n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 7.8 Ki ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
O96013 PAK4 Homo sapiens Human PF00786 PF00069 6.2 Ki ChEMBL;BindingDB