Molecule Details
InChIKeyGHZDTANYDBSHNU-IOZNDOSASA-N
Compound NameN-alpha-Ac-[Ala26,Phe27]PYY(22-36)-NH2(N-alpha-Ac-ASLAAFLNLVTRQRY-NH2)
Canonical SMILESCC(=O)N[C@@H](C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)[C@@H](C)O)C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49146 NPY2R Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P25929 NPY1R Homo sapiens Human PF00001 6.2 IC50 ChEMBL;BindingDB