Molecule Details
InChIKeyGHWRYTXWRJFGJW-UHFFFAOYSA-N
Compound Name6-chloro-5-fluoro-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl)indoline-1-carboxamide
Canonical SMILESCc1ncccc1Oc1ccc(NC(=O)N2CCc3cc(F)c(Cl)cc32)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB