Molecule Details
InChIKeyGHDKYBCUDPSXGJ-UHFFFAOYSA-N
Compound Name4-((3-Bromo-4-O-sulfamoylbenzyl)(4-cyanophenyl)amino)-4H-(1,2,4)-triazole
Canonical SMILESN#Cc1ccc(N(Cc2ccc(OS(N)(=O)=O)c(Br)c2)n2cnnc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.79
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB04600
Drug Name4-[(3-BROMO-4-O-SULFAMOYLBENZYL)(4-CYANOPHENYL)AMINO]-4H-[1,2,4]-TRIAZOLE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 10020 CHEMBL108483 ChemSpider: 3571981 PDB: 4TR PubChem:4369414 PubChem:46508682 ZINC: ZINC000003991718
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11511 CYP19A1 Homo sapiens Human PF00067 9.1 IC50 ChEMBL;BindingDB
P08842 STS Homo sapiens Human PF00884 PF14707 7.4 IC50 ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.9 IC50 BindingDB
DrugBank Target Actions (1)
Target Gene Target Name Action Type
P00918 CA2 Carbonic anhydrase 2 binder targets