Molecule Details
InChIKeyGHAZMUIBGZEWFT-UHFFFAOYSA-N
Compound Name4-[(3,5-dimethyl-1-adamantyl)carbamoylamino]-3-fluoro-N-[6-(hydroxyamino)-6-oxohexyl]benzamide
Canonical SMILESCC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCC(=O)NO)cc1F)(C3)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.5
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P34913 EPHX2 Homo sapiens Human PF00561 PF00702 9.3 IC50 ChEMBL
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.3 IC50 ChEMBL
O15379 HDAC3 Homo sapiens Human PF00850 7.3 IC50 ChEMBL
Q92769 HDAC2 Homo sapiens Human PF00850 6.1 IC50 ChEMBL