Molecule Details
InChIKeyGGLRFXACWCOWSX-UHFFFAOYSA-N
Compound NameN-[(6-pyrrolidin-1-yl-3-pyridinyl)methyl]-2-[[4-(trifluoromethoxy)phenyl]methyl]-1,3-oxazole-4-carboxamide
Canonical SMILESO=C(NCc1ccc(N2CCCC2)nc1)c1coc(Cc2ccc(OC(F)(F)F)cc2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.3 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 7.7 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.5 IC50 ChEMBL;BindingDB