Molecule Details
InChIKeyGGKUJNMJJNAMPQ-UHFFFAOYSA-N
Compound NameN-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1,2,3,4-tetrahydroquinolin-3-yl]-(1-methyl-1H-imidazole-4-sulfonyl)amino]acetamide
Canonical SMILESCn1cnc(S(=O)(=O)N(CC(=O)NC(C)(C)C)C2Cc3cc(C#N)ccc3N(Cc3cncn3C)C2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.92
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5E175 rhlE Aliivibrio fischeri (strain ATCC 700601 / ES114) Pathogen PF00270 PF00271 8.9 IC50 BindingDB
Q5EI73 Plasmodium falciparum Pathogen PF01239 8.9 IC50 ChEMBL