Molecule Details
InChIKeyGFQVWAVVNKSCBU-UHFFFAOYSA-N
Compound Name5-[4-[4-(2-fluoroanilino)quinazolin-6-yl]triazol-1-yl]-N-hydroxypentanamide
Canonical SMILESO=C(CCCCn1cc(-c2ccc3ncnc(Nc4ccccc4F)c3c2)nn1)NO
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.44
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 9.0 IC50 ChEMBL
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 8.4 IC50 ChEMBL
P00533 EGFR Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 8.0 IC50 ChEMBL