Molecule Details
InChIKeyGFBYPYUSXALYJS-UHFFFAOYSA-N
Compound Name2-[2-(Cyclopropanecarbonylamino)-4-pyridinyl]-4-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethoxy]-1,3-thiazole-5-carboxylic acid
Canonical SMILESO=C(O)c1sc(-c2ccnc(NC(=O)C3CC3)c2)nc1OCCNc1c2c(nc3ccccc13)CCCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 6.3 IC50 ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 6.2 IC50 ChEMBL;BindingDB