Molecule Details
InChIKeyGEUNWTZTVWNSTN-UHFFFAOYSA-N
Compound NameN-{4-[1-(3-Hydroxypropyl)-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}-N''-phenylurea
Canonical SMILESO=C(Nc1ccccc1)Nc1ccc(-c2nn(CCCO)cc2-c2ccnc3[nH]ccc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.91
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.0 pIC50 TTD_MultiTarget