Molecule Details
InChIKeyGEOWQTGMJLRVOC-HHHXNRCGSA-N
Compound Name1-{1-((R)-Benzyloxymethyl)-2-[4-(4-fluoro-benzoyl)-piperidin-1-yl]-2-oxo-ethyl}-3-m-tolyl-urea
Canonical SMILESCc1cccc(NC(=O)N[C@H](COCc2ccccc2)C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.64
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.6 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.6 IC50 ChEMBL;BindingDB