Molecule Details
InChIKeyGEDMTUQQRHRNSK-UHFFFAOYSA-N
Compound NameN-[4-[(5-methoxy-3,4-dihydro-2H-chromen-3-yl)-propylamino]butyl]-4-oxo-3-oxa-13-azatetracyclo[7.7.1.02,7.013,17]heptadeca-1(17),2(7),5,8-tetraene-6-carboxamide
Canonical SMILESCCCN(CCCCNC(=O)c1cc(=O)oc2c3c4c(cc12)CCCN4CCC3)C1COc2cccc(OC)c2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 9.5 IC50 BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.1 IC50 BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.8 IC50 BindingDB