Molecule Details
InChIKeyGDZTURHUKDAJGD-UHFFFAOYSA-N
Compound Name4-[4-(2,4-Dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]phenol
Canonical SMILESCc1nc(C)c(-c2ccnc(Nc3ccc(O)cc3)n2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.85
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget