Molecule Details
InChIKeyGDHDKBHKLQDVFR-UHFFFAOYSA-N
Compound Namebutyl N-[2-[4-[[2-ethyl-6-(morpholine-4-carbonylamino)-4-oxoquinazolin-3-yl]methyl]-3-fluorophenyl]phenyl]sulfonylcarbamate
Canonical SMILESCCCCOC(=O)NS(=O)(=O)c1ccccc1-c1ccc(Cn2c(CC)nc3ccc(NC(=O)N4CCOCC4)cc3c2=O)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P50052 AGTR2 Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB
P30556 AGTR1 Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB