Molecule Details
InChIKeyGCTSHJXOIFKTDC-UHFFFAOYSA-N
Canonical SMILESCOc1ccc2c(c1Nc1cccc(C(F)(F)F)c1)CN(C#N)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.56
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15561 TEAD4 Homo sapiens Human PF01285 PF17725 6.6 IC50 ChEMBL
P28347 TEAD1 Homo sapiens Human PF01285 PF17725 6.5 IC50 ChEMBL