Molecule Details
InChIKeyGCKBOFRETXSMFP-ACCUITESSA-N
Compound Name1-phenyl-N-(3-styryl-1H-indazol-5-yl)methanesulfonamide
Canonical SMILESO=S(=O)(Cc1ccccc1)Nc1ccc2[nH]nc(/C=C/c3ccccc3)c2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.48
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.5 pIC50 TTD_MultiTarget