Molecule Details
InChIKeyGCIMHCJOZUYMTH-UHFFFAOYSA-N
Compound Name3-[[4-[2-(3-Oxa-8-azabicyclo[3.2.1]octan-8-yl)-4-pyridinyl]pyrimidin-2-yl]amino]benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1cccc(Nc2nccc(-c3ccnc(N4C5CCC4COC5)c3)n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96Q15 SMG1 Homo sapiens Human PF02260 PF00454 PF15785 PF17229 7.6 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB