Molecule Details
InChIKeyGCFCQBCBKXQUCD-UHFFFAOYSA-N
Compound Name1-methyl-8-(2-(trifluoromethoxy)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Canonical SMILESCn1nc(C(N)=O)c2c1-c1nc(Nc3ccccc3OC(F)(F)F)ncc1CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H4B4 PLK3 Homo sapiens Human PF00069 PF00659 7.5 IC50 ChEMBL;BindingDB
P53350 PLK1 Homo sapiens Human PF00069 PF00659 6.9 IC50 ChEMBL;BindingDB
Q9NYY3 PLK2 Homo sapiens Human PF00069 PF00659 6.7 IC50 ChEMBL;BindingDB