Molecule Details
InChIKeyGBXVVXZXFOFHSU-UHFFFAOYSA-N
Compound NameN-(4-(4-(5-methyl-1H-pyrazol-3-ylamino)-6-(pyridin-3-yl)pyrimidin-2-ylthio)phenyl)propionamide
Canonical SMILESCCC(=O)Nc1ccc(Sc2nc(Nc3cc(C)[nH]n3)cc(-c3cccnc3)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.03
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 Ki ChEMBL;BindingDB