Molecule Details
InChIKeyGBRORGYPYNNDGL-UHFFFAOYSA-N
Compound Name1-(Dimethylamino)-3-(4-(4-(6-morpholinopyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-ylamino)phenoxy)propan-2-ol
Canonical SMILESCN(C)CC(O)COc1ccc(Nc2nccc(-c3cnn4nc(N5CCOCC5)ccc34)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.64
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.3 pIC50 TTD_MultiTarget
P49841 GSK3B Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB