Molecule Details
InChIKeyGBQAIAULXOPTMN-FLNNQWSLSA-N
Compound Name(1R,2S,6R,8S)-4,4,11,11-tetramethyl-N-sulfamoyl-3,5,7,10,12-pentaoxatricyclo[6.4.0.02,6]dodecane-6-carboxamide
Canonical SMILESCC1(C)OC[C@@H]2O[C@@]3(C(=O)NS(N)(=O)=O)OC(C)(C)O[C@H]3[C@@H]2O1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.82
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.2 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.2 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB