Molecule Details
InChIKeyGBKQNVNYZATRQE-UHFFFAOYSA-N
Compound Name4-(8-aminonaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Canonical SMILESNc1cccc2ccc(-n3c(-c4ccnc(NC5CCOCC5)c4)n[nH]c3=O)cc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.63
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB