Molecule Details
InChIKeyGAMJJHMLLXIWRZ-OCCSQVGLSA-N
Compound Nametert-butyl N-[(3S,6R)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl]carbamate
Canonical SMILESC[C@@H]1CC[C@H](NC(=O)OC(C)(C)C)CN1c1cc(-c2ccc3c(N)n[nH]c3c2)nc(N)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 7.3 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 6.2 IC50 ChEMBL;BindingDB