Molecule Details
InChIKeyFZWFQSYPXVHFDQ-KPKJPENVSA-N
Compound Name4-[(2,6-dimethoxybenzoyl)amino]-N-[1-[3-[[(E)-4-(dimethylamino)but-2-enoyl]amino]phenyl]sulfonylpiperidin-4-yl]-1H-pyrazole-5-carboxamide
Canonical SMILESCOc1cccc(OC)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCN(S(=O)(=O)c2cccc(NC(=O)/C=C/CN(C)C)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.54
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00536 CDK16 Homo sapiens Human PF00069 8.0 IC50 BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.6 IC50 BindingDB
O94921 CDK14 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
Q8ND76 CCNY Homo sapiens Human PF00134 7.3 IC50 ChEMBL