Molecule Details
InChIKeyFZPWJZCQBCBZKE-UHFFFAOYSA-N
Canonical SMILESCc1ccc(Nc2ncc3c(n2)N(C)C(=O)N(c2cc(NC(=O)c4ccc(CN5CCN(C)CC5)c(C(F)(F)F)c4)ccc2C)C3)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12851 MAP4K2 Homo sapiens Human PF00780 PF00069 8.3 IC50 ChEMBL;BindingDB
Q07912 TNK2 Homo sapiens Human PF09027 PF11555 PF07714 PF22931 PF14604 7.6 IC50 ChEMBL;BindingDB