Molecule Details
InChIKeyFZMCQVGUQKFBIJ-CYBMUJFWSA-N
Compound Name4-(3-methylanilino)-2-[[(3R)-piperidin-3-yl]amino]pyrimidine-5-carboxamide
Canonical SMILESCc1cccc(Nc2nc(N[C@@H]3CCCNC3)ncc2C(N)=O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43405 SYK Homo sapiens Human PF07714 PF00017 6.9 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 6.8 IC50 ChEMBL
P28482 MAPK1 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB