Molecule Details
InChIKeyFYMYEYOPWYBNKY-UHFFFAOYSA-N
Canonical SMILESO=C(Nc1ccc2[nH]cc(C3CCN(Cc4cccc(CN5CCC(c6c[nH]c7ccc(NC(=O)c8ccc(F)cc8)cc67)CC5)c4)CC3)c2c1)c1ccc(F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB