Molecule Details
InChIKeyFXRXKUVQNAIPQC-KXUCPTDWSA-N
Compound Name(2S)-2-[[(2S,5R)-2-(acetamidomethylcarbamoyl)-3-methyl-7-oxo-1,6-diazabicyclo[3.2.1]oct-3-en-6-yl]oxy]-2-fluoroacetic acid
Canonical SMILESCC(=O)NCNC(=O)[C@@H]1C(C)=C[C@@H]2CN1C(=O)N2O[C@@H](F)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.71
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00811 ampC Escherichia coli (strain K12) Pathogen PF00144 8.5 IC50 ChEMBL;BindingDB
Q6XEC0 OXA-48 Klebsiella pneumoniae Pathogen PF00905 7.3 IC50 BindingDB
P62593 bla Escherichia coli Pathogen PF13354 7.3 IC50 BindingDB