Molecule Details
InChIKeyFXMBSEOFWALADX-UHFFFAOYSA-N
Compound Name4-[5-[1-(Oxetan-3-yl)pyrazol-4-yl]-3-pyridinyl]-2-propan-2-yloxybenzamide
Canonical SMILESCC(C)Oc1cc(-c2cncc(-c3cnn(C4COC4)c3)c2)ccc1C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HBH9 MKNK2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P06730 EIF4E Homo sapiens Human PF01652 6.7 IC50 ChEMBL
Q9BUB5 MKNK1 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB