Molecule Details
InChIKeyFXBNFLKLXHFULB-UHFFFAOYSA-N
Compound NameN-(4-bromo-3-(1H-1,2,4-triazol-3-yl)thiophen-2-yl)-2-(3-(trifluoromethyl)quinolin-5-yl)acetamide
Canonical SMILESO=C(Cc1cccc2ncc(C(F)(F)F)cc12)Nc1scc(Br)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB