Molecule Details
InChIKeyFWXRRJODQJLGKY-UHFFFAOYSA-N
Compound Name8-[(6-Carbamoyl-3-pyridinyl)oxy]-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
Canonical SMILESNC(=O)c1ccc(Oc2sc(C(N)=O)c3c2-c2sncc2CC3)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 9.0 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 9.0 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB