Molecule Details
InChIKeyFWQGDGPDBUUACD-OKDNLZPVSA-N
Compound Name(2S,5S,8R,11R)-5-[3-(diaminomethylideneamino)propyl]-8-(1H-indol-3-ylmethyl)-2-(naphthalen-2-ylmethyl)-3,6,9,16,19-pentaoxo-1,4,7,10,15-pentazacyclononadecane-11-carboxamide
Canonical SMILESN=C(N)NCCC[C@@H]1NC(=O)[C@H](Cc2ccc3ccccc3c2)NC(=O)CCC(=O)NCCC[C@H](C(N)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB