Molecule Details
InChIKeyFVOXTVYJOXVETI-VKVKMMGJSA-N
Compound Name4-[4-[(Z)-[[4-(6-bromo-2-oxochromen-3-yl)-1,3-thiazol-2-yl]hydrazinylidene]methyl]-3-(4-fluorophenyl)pyrazol-1-yl]benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1ccc(-n2cc(/C=N\Nc3nc(-c4cc5cc(Br)ccc5oc4=O)cs3)c(-c3ccc(F)cc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 8.3 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.7 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB