Molecule Details
InChIKeyFVNNTRZFDXTUGO-UHFFFAOYSA-N
Compound Name2-[2-[(4,5-Difluoro-2-methylphenoxy)methyl]-5-methoxy-4-pyridinyl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one
Canonical SMILESCOc1cnc(COc2cc(F)c(F)cc2C)cc1-c1cc2c([nH]1)CCNC2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P78368 CSNK1G2 Homo sapiens Human PF12605 PF00069 7.4 IC50 ChEMBL;BindingDB
P48730 CSNK1D Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P48729 CSNK1A1 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB