Molecule Details
InChIKeyFVIKWIZJEHFVFM-JOMNFKBKSA-N
Compound Name2-[3-[(2S,4R)-6-carbamimidoyl-4-phenyl-1,2,3,4-tetrahydroquinolin-2-yl]phenyl]-5-(2-methylpropylcarbamoyl)benzoic acid
Canonical SMILESCC(C)CNC(=O)c1ccc(-c2cccc([C@@H]3C[C@H](c4ccccc4)c4cc(C(=N)N)ccc4N3)c2)c(C(=O)O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 7.6 Ki ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.6 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.6 Ki ChEMBL