Molecule Details
InChIKeyFVFURMJFTAJXRH-UHFFFAOYSA-N
Compound NameN-(1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl)-7-fluoro-4-oxo-4H-chromene-2-carboxamide
Canonical SMILESO=C(NC1CCN(Cc2ccc3c(c2)OCO3)CC1)c1cc(=O)c2ccc(F)cc2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99705 MCHR1 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 7.8 IC50 ChEMBL;BindingDB
Q969V1 MCHR2 Homo sapiens Human PF00001 7.5 IC50 ChEMBL