Molecule Details
InChIKeyFUGFIYPWJLQXJO-UHFFFAOYSA-N
Compound Name6-[[2-methoxy-N-methyl-5-(trifluoromethyl)anilino]methyl]-5-methyl-pyrido[2,3-d]pyrimidine-2,4-diamine
Canonical SMILESCOc1ccc(C(F)(F)F)cc1N(C)Cc1cnc2nc(N)nc(N)c2c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 7.4 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 8.9 IC50 ChEMBL
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.4 IC50 ChEMBL;BindingDB