Molecule Details
InChIKeyFUBBWDWIGBTUPQ-UHFFFAOYSA-N
Compound NameAxitirome
Canonical SMILESCCOC(=O)C(=O)Nc1cc(C)c(Oc2ccc(O)c(C(O)c3ccc(F)cc3)c2)c(C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10828 THRB Homo sapiens Human PF00104 PF00105 8.7 Ki ChEMBL;BindingDB
P10827 THRA Homo sapiens Human PF00104 PF00105 7.4 Ki ChEMBL;BindingDB